Growth Hormone Antagonist Therapies for Neurological Disorders and Veterinary Applications

Publication ID: 24-11857602_0002_PTD
Published: October 28, 2025
Category:New Applications & Use Cases

Legal Citation

pr1or.art Inc., “Growth Hormone Antagonist Therapies for Neurological Disorders and Veterinary Applications,” Published Technical Disclosure No. 24-11857602_0002_PTD, Published October 28, 2025, available at https://archive.pr1or.art/24-11857602_0002_PTD
This technical disclosure describes improvements that would be readily apparent to a Person Having Ordinary Skill In The Art (PHOSITA) when considered in combination with the foundational architecture disclosed in U.S. Patent No. 11,857,602.

Summary of the Inventive Concept

This inventive concept leverages the core technology of the original patent to develop novel therapies for neurological disorders, veterinary applications, and age-related diseases, expanding the scope of growth hormone antagonist treatments beyond cancer.

Background and Problem Solved

The original patent disclosed a composition for treating cancer and other diseases using a human growth hormone receptor antagonist. However, there remains a need for effective treatments for neurological disorders, veterinary applications, and age-related diseases. This inventive concept addresses these limitations by exploring new applications and use cases for the core technology.

Detailed Description of the Inventive Concept

The new claims describe methods and systems for treating neurological disorders, delivering growth hormone receptor antagonists to target sites, and preventing or treating age-related diseases. These innovative approaches involve conjugating the antagonist with polyethylene glycol molecules, using microneedle arrays for transdermal delivery, and modifying the antagonist for increased efficacy against canine or feline cancers.

Novelty and Inventive Step

The new claims introduce novel and non-obvious applications of the growth hormone receptor antagonist technology, expanding its scope beyond cancer treatment and into new therapeutic areas. The inventive step lies in the identification of new uses and modifications that enable the antagonist to address unmet needs in neurological disorders, veterinary applications, and age-related diseases.

Alternative Embodiments and Variations

Alternative embodiments of the inventive concept could include using different polyethylene glycol molecules, modifying the antagonist for use in other diseases or conditions, or developing new formulations for oral or injectable delivery. Variations of the microneedle array design could also be explored to optimize transdermal delivery.

Potential Commercial Applications and Market

The inventive concept has significant commercial potential in the pharmaceutical and biotechnology industries, particularly in the areas of neurological disorders, veterinary medicine, and age-related diseases. The market for these applications is substantial, with a growing need for effective treatments and therapies.

CPC Classifications

SectionClassGroup
A A61 A61K38/27
A A61 A61K45/06
A A61 A61K47/10
A A61 A61P35/00
A A61 A61K2039/505

Field of Art

Biotechnology and pharmaceutical sciences, specifically focusing on protein engineering, receptor antagonists, and targeted therapeutic compositions for cancer and neurological disorders

Person of Ordinary Skill (PHOSITA) Profile

A researcher with advanced degree in molecular biology or biochemistry, experienced in protein modification, drug delivery systems, and receptor-based therapeutic strategies, familiar with conjugation techniques and drug formulation approaches

Obviousness Rationale

A person having ordinary skill would recognize that the source patent's growth hormone receptor antagonist technology provides a foundational platform for exploring alternative therapeutic applications. The PTD's variations represent predictable extensions of the original patent's core technology by applying known protein engineering and drug delivery techniques to expand treatment modalities. The modifications demonstrate standard approaches in pharmaceutical research for optimizing drug delivery, targeting new disease states, and improving therapeutic efficacy.

Obvious Combinations & Variations

Source Patent Element
Growth hormone receptor antagonist with specific amino acid substitutions
PTD Variation
Modifying antagonist for veterinary cancer treatments in canine and feline applications
Obviousness Reasoning
Routine protein engineering technique to adapt molecular structures for species-specific targeting, representing a predictable variation within known protein modification strategies
Source Patent Element
Polyethylene glycol conjugation with maleimide group
PTD Variation
Using microneedle array for transdermal delivery of PEG-conjugated antagonist
Obviousness Reasoning
Combining known drug delivery technologies represents an obvious optimization approach, applying standard pharmaceutical formulation techniques to improve drug administration
Source Patent Element
Cancer treatment composition with growth hormone receptor antagonist
PTD Variation
Expanding treatment to neurological disorders and age-related conditions
Obviousness Reasoning
Exploring alternative therapeutic applications for a known molecular mechanism is a standard scientific approach, representing a predictable extension of existing research
Source Patent Element
Antagonist with specific receptor interaction properties
PTD Variation
Developing biosensor monitoring system for tracking antagonist efficacy
Obviousness Reasoning
Creating diagnostic tools to monitor therapeutic interventions is a routine approach in pharmaceutical research, representing an obvious technological progression
35 U.S.C. § 103 Summary: Based on the teachings of US Patent 11857602, the disclosed variations in therapeutic applications, delivery methods, and molecular modifications of growth hormone receptor antagonists would have been obvious to a person having ordinary skill in the art at the time of invention. The predictable combination of known protein engineering techniques, drug delivery strategies, and expanded therapeutic targeting renders the claimed innovations prima facie obvious under 35 U.S.C. ยง 103.

Original Patent Information

Patent NumberUS 11,857,602
TitleGrowth hormone antagonist and anti-cancer composition combination therapy